New Quinoline Analogues: As Potential Diabetics Inhibitors and Molecular Docking Study
The 7-quinolinyl bearing 1,3,4-thiadiazole-2-amine analogues were synthesized (1–17) and based on the literature these analog were screened in vitro for their α-amylase and α-glucosidase inhibitory profile. All analogues showed moderate to good inhibitory potentials ranging between 0.80 ± 0.05 µM to...
Published in: | Polycyclic Aromatic Compounds |
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Main Author: | Taha M.; Salahuddin M.; Rahim F.; Imran S.; Hussain S.; Uddin N.; Khan K.M. |
Format: | Article |
Language: | English |
Published: |
Taylor and Francis Ltd.
2024
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Online Access: | https://www.scopus.com/inward/record.uri?eid=2-s2.0-85147419609&doi=10.1080%2f10406638.2023.2169471&partnerID=40&md5=cb67df0ec9786609431d71c436d8e0ce |
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