New thiazole-based thiazolidinone derivatives: Synthesis, in vitro α-amylase, α-glucosidase activities and silico molecular docking study
A series of thiazole-based thiazolidinone derivatives (1-20) have been synthesized and evaluated against α-glucosidase and α-amylase enzymes. All derivatives showed good α-glucosidase activity having IC50 values ranging from 2.40 ± 0.10 to 31.40 ± 0.90 μM and for α-amylase having IC50 values ranging...
Published in: | Chemical Data Collections |
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Main Author: | Khan S.; Ullah H.; Rahim F.; Taha M.; Hussain R.; Khan M.S.; Ali H.; Khan M.U.; Shah S.A.A.; Khan K.M. |
Format: | Data paper |
Language: | English |
Published: |
Elsevier B.V.
2022
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Online Access: | https://www.scopus.com/inward/record.uri?eid=2-s2.0-85142669443&doi=10.1016%2fj.cdc.2022.100967&partnerID=40&md5=3d2e0201d96f4b145daa5366ea80f3bc |
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