Bacterial Biofilm Inhibition, Hemolytic Activity, and Structure–Activity Relationship of N-(2,3-Dihydro-1,4-Benzodioxin-6-yl)-4-Nitro-N-(Substituted-Benzyl)benzenesulfonamides

QR Code

Bacterial Biofilm Inhibition, Hemolytic Activity, and Structure–Activity Relationship of N-(2,3-Dihydro-1,4-Benzodioxin-6-yl)-4-Nitro-N-(Substituted-Benzyl)benzenesulfonamides

Abstract: In the work, new antibacterial compounds that combine sulfonamide and benzodioxane fragments in their framework were fabricated. Structures of the sulfonamide derivatives were determined by the IR, 1H NMR, 13C NMR, and EI-MS spectroscopy techniques. Antibacterial potential of these molecul...

Full description

Bibliographic Details
Published in:	Russian Journal of Bioorganic Chemistry
Main Author:	2-s2.0-85083967679
Format:	Article
Language:	English
Published:	Pleiades Publishing 2020
Online Access:	https://www.scopus.com/inward/record.uri?eid=2-s2.0-85083967679&doi=10.1134%2fS1068162020020028&partnerID=40&md5=58d8204571e91024f097916229c5f6da

Similar Items

Synthesis, Bacterial biofilm inhibition and cytotoxicity of new N-Alkyl/aralkyl-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-nitrobenzenesulfonamides
by: 2-s2.0-85077925901
Published: (2020)

Synthesis of some new N-substituted-N-(2,3-Dihydro-[1,4]benzodioxin-6-yl)-4-acetamidobenzenesulfonamides as valuable antibacterial agents
by: 2-s2.0-84962661129
Published: (2016)

Synthesis of Some New N-Alkyl/Aralkyl-N-(2,3-Dihydro-1,4-Benzodioxin-6-YL)-4-Bromobenzenesulfonamides as Possible Therapeutic Agents F or Alzheimer’s Disease
by: 2-s2.0-85127408369
Published: (2022)

Synthesis, antibacterial and lipoxygenase inhibition studies of N-(Alkyl/aralkyl)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-methylbenzenesulfonamides; [N-(Alkil/aralkil)-N-(2,3-dihidro-1,4-benzodioksin-6-il)-4-metilbenzensülfonamitlerin Sentezi ile Antibakteriyel ve Lipoksijenaz İnhibitör Özellikleri]
by: 2-s2.0-85013177487
Published: (2017)

Synthesis of 2-[2,3-dihydro-1,4-benzodioxin-6-yl(phenylsulfonyl)amino]-N-(un/substitutedphenyl)acetamides as anti-diabetic agents
by: 2-s2.0-85143584454
Published: (2022)

Synthesis of promising antibacterial and antifungal agents: 2-[[(4-Chlorophenyl)sulfonyl](2,3-dihydro-1,4-benzodioxin-6-yl)amino]-N(un/substituted-phenyl)acetamides
by: 2-s2.0-85091220218
Published: (2020)

Synthesis, bacterial biofilm inhibition and hemolytic activity of 4-chloro-n-(dimethylphenyl)butamide regio-isomers
by: 2-s2.0-85100876566
Published: (2020)

Synthesis of new 2-{2,3-dihydro-1,4-benzodioxin-6-yl[(4‑methylphenyl) sulfonyl]amino}-N-(un/substituted-phenyl) acetamides as α-glucosidase and acetylcholinesterase inhibitors and their in silico study
by: 2-s2.0-85073287972
Published: (2019)

Synthesis of novel N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-{[5-(un/substituted-phenyl)-1,3,4-oxadiazol-2-yl]sulfanyl}acetamides as potent antibacterial agents
by: 2-s2.0-85129100563
Published: (2022)

Synthesis of some new N-(alkyl/aralkyl)-N-(2,3-dihydro-1,4-benzodioxan-6-yl)-4-chlorobenzenesulfonamides as possible therapeutic agents for Alzheimer’s disease and Type-2 Diabetes
by: 2-s2.0-85061745776
Published: (2019)

Synthesis, characterization, antibacterial, α-glucosidase inhibition and hemolytic studies on some new n-(2,3-Dimethylphenyl)benzenesulfonamide derivatives
by: 2-s2.0-84962385188
Published: (2016)

Synthetic N-aralkylated-N-(2,4-dimethylphenyl)benzenesulfonamides: As potent anti-bacterial agents
by: 2-s2.0-85009833752
Published: (2016)

Synthesis of some new N-(alkyl/aralkyl)-N-(4-methoxyphenethyl) benzenesulfonamides as antibacterial agents against Escherichia coli
by: 2-s2.0-85072317017
Published: (2019)

Synthesis, characterization, antibacterial, hemolytic and thrombolytic activity evaluation of 5-(3-chlorophenyl)-2-((N-(substituted)-2-acetamoyl)sulfanyl)-1,3,4-oxadiazole derivatives
by: 2-s2.0-85090106052
Published: (2020)

N-([1,1ʹ-biaryl]-4-yl)-1-naphthamide-based scaffolds synthesis, their cheminformatics analyses, and screening as bacterial biofilm inhibitor
by: 2-s2.0-85118291164
Published: (2022)

Efficient synthesis of 2,3-diarylbenzo[b]thiophene molecules through palladium (0) Suzuki–Miyaura cross-coupling reaction and their antithrombolyitc, biofilm inhibition, hemolytic potential and molecular docking studies
by: 2-s2.0-85085920123
Published: (2020)

Nanostructured materials based on g-C3N4 for enhanced photocatalytic activity and potentials application: A review
by: Sohail M.; Anwar U.; Taha T.A.; Qazi H.I.A.; Al-Sehemi A.G.; Ullah S.; Algarni H.; Ahmed I.M.; Amin M.A.; Palamanit A.; Iqbal W.; Alharthi S.; Nawawi W.I.; Ajmal Z.; Ali H.; Hayat A.
Published: (2022)

Synthesis of N-substituted acetamide derivatives of azinane-bearing 1,3,4-oxadiazole nucleus and screening for antibacterial activity
by: 2-s2.0-85014071417
Published: (2017)

Synthesis, enzyme inhibitory kinetics mechanism and computational study of N-(4-methoxyphenethyl)-N-(substituted)- 4-methylbenzenesulfonamides as novel therapeutic agents for Alzheimer's disease
by: 2-s2.0-85049259205
Published: (2018)

Synthesis and in silico study of 2-furyl(4-{4-[(substituted)sulfonyl]benzyl}-1-piperazinyl)methanone derivatives as suitable therapeutic agents
by: Hussain G.; Abbasi M.A.; Aziz-ur-Rehman; Siddiqui S.Z.; Shah S.A.A.; Ashraf M.; Qurat-ul-Ain; Ahmad I.; Malik R.; Lodhi M.A.; Khan F.A.; Shahid M.; Fatima H.
Published: (2017)

Synthesis and in silico study of 2-furyl(4-{4-[(substituted)sulfonyl]benzyl}-1-piperazinyl)methanone derivatives as suitable therapeutic agents
by: 2-s2.0-85018664413
Published: (2017)

Facile synthesis and characterization of a visible light-active ternary TiO2/ZnS/g-C3N4 heterostructure for multipollutant degradation
by: Kanakaraju, et al.
Published: (2024)

Α-Glucosidase inhibitory potential and hemolytic evaluation of newly synthesized 3, 4, 5-trisubstituted-1, 2, 4-triazole derivatives
by: 2-s2.0-85077924129
Published: (2019)

Ultrafast laser plasma doping of Er3+ in Si3N4-on-silicon
by: Kamil S.A.; Chandrappan J.; Krauss T.F.; Jose G.
Published: (2019)

Synthesis, spectral analysis and biological evaluation of N-alkyl/aralkyl/aryl-4-chlorobenzenesulfonamide derivatives
by: 2-s2.0-84989919539
Published: (2016)

Novel isoxazolinyl spiropyrrolidinediones: 1,3-dipolar cycloaddition of 1-benzyl-3,3-dimethyl-5-methylenepyrrolidin-2,4-dione
by: Bathich Y.; Syed Monudeen Khan S.E.B.; Hamzah A.S.
Published: (2011)

Synthesis, enzyme inhibitory kinetics, & computational studies of N-(substituted phenyl)-(5-(3,4-dichlorobenzyl)-4-(4-chlorophenyl)-4H-1,2,4-triazol-3-ylthio)methylbenzamides: As potent alkaline phosphatase inhibitors
by: 2-s2.0-85204404556
Published: (2025)

Synergistic Antibacterial Screening of Cymbopogon citratus and Azadirachta indica: Phytochemical Profiling and Antioxidant and Hemolytic Activities
by: 2-s2.0-85159588072
Published: (2023)

Design, synthesis of triazole-based scaffolds, N-(substitutedphenyl)-2-(5-(4-methoxyphenyl)-4-phenyl-4H-1,2,4-triazol-3-ylthiol)acetamides: As potential anti-cholinesterase agents for neurodegenerative diseases
by: 2-s2.0-85160806262
Published: (2023)

Synthesis, spectral analysis and pharmacological study of N’-substituted-2-(5-((2,4-dimethylphenoxy)methyl)-1,3,4-oxadiazol-2-ylthio)acetohydrazides
by: 2-s2.0-85006043172
Published: (2016)

Synthesis, in vitro antimicrobial, anticancer evaluation and QSAR studies of N'-(substituted)-4-(butan-2-lideneamino)benzohydrazides
by: 2-s2.0-84905580114
Published: (2014)

Designing, Synthesis and Characterization of Fluorescent Fluorescein Hydrazides and Antibacterial Studies against Sinusitis Isolates and Hemolytic Activities
by: Kousar, et al.
Published: (2024)

Designing, Synthesis and Characterization of Fluorescent Fluorescein Hydrazides and Antibacterial Studies against Sinusitis Isolates and Hemolytic Activities
by: 2-s2.0-86000365896
Published: (2024)

Ethyl 4-[(2-hydroxyethyl)amino]-2-(4-methoxy-phenyl)-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxylate
by: Abdul Rashid F.N.A.; Mohammat M.F.; Abdul Manan M.A.F.; Bakhtiar Afendy A.A.A.; Cordes D.B.; McKay A.P.
Published: (2024)

Recent Advancement of the Current Aspects of g-C3N4 for its Photocatalytic Applications in Sustainable Energy System
by: Hayat A.; Sohail M.; Ali Shah Syed J.; Al-Sehemi A.G.; Mohammed M.H.; Al-Ghamdi A.A.; Taha T.A.; Salem AlSalem H.; Alenad A.M.; Amin M.A.; Palamanit A.; Liu C.; Nawawi W.I.; Tariq Saeed Chani M.; Muzibur Rahman M.
Published: (2022)

Synthesis, Kinetics and Computational Explorations of 4-Phenylpiperazine Bearing N-(Aryl)-3-substituted-benzamides as Auspicious Tyrosinase Inhibitors
by: 2-s2.0-85187520882
Published: (2024)

Efficient Synthesis of 4-Bromo-N-(1-phenylethyl)benzamide, Arylation by Pd(0) Catalyst, Characterization and DFT Study
by: 2-s2.0-85135826802
Published: (2022)

Recent Advancement of the Current Aspects of g-C3N4 for its Photocatalytic Applications in Sustainable Energy System
by: 2-s2.0-85124751328
Published: (2022)

Surface Physicochemistry Modification and Structural Nanoarchitectures of g-C3N4 for Wastewater Remediation and Solar Fuel Generation
by: 2-s2.0-85122536288
Published: (2022)

Graphitic carbon nitride (g–C3N4)–based semiconductor as a beneficial candidate in photocatalysis diversity
by: 2-s2.0-85121209781
Published: (2022)