Synthesis, kinetics, binding conformations and structure-activity relationship of potent tyrosinase inhibitors: Aralkylated 2-aminothiazole-ethyltriazole hybrids

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Synthesis, kinetics, binding conformations and structure-activity relationship of potent tyrosinase inhibitors: Aralkylated 2-aminothiazole-ethyltriazole hybrids

Considering the diversified pharmacological importance of thiazole and triazole heterocyclic moieties, a unique series of S-aralkylated bi-heterocyclic hybrids, 7a-l, was synthesized in a convergent manner. The structures of newly synthesized compounds were characterized by 1 H-NMR,13C-NMR, IR, and...

وصف كامل

التفاصيل البيبلوغرافية
الحاوية / القاعدة:	Iranian Journal of Pharmaceutical Research
المؤلف الرئيسي:	2-s2.0-85111424369
التنسيق:	مقال
اللغة:	English
منشور في:	Iranian Journal of Pharmaceutical Research 2021
الوصول للمادة أونلاين:	https://www.scopus.com/inward/record.uri?eid=2-s2.0-85111424369&doi=10.22037%2fijpr.2020.15521.13145&partnerID=40&md5=fac8f033ad621c698eed9be97fe4926b

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