Discovering biological efficacy of new thiadiazole as effective inhibitors of urease, glycation, and (DPPH) scavengers: Biochemical and in silico study
Thiadiazole is a potential class of α-glucosidase, β-glucuronidase, and anti-leishmanial inhibitors. Our aim was to develop thiadiazole based dual inhibitors for urease glycation inhibition and (DDPH) scavenging activity. Pyridine-based-thiadiazole analogs (1–18) were synthesized and characterized t...
Published in: | Journal of Molecular Structure |
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Main Author: | Taha M.; Imran S.; Rahim F.; Uddin N.; Iqbal N.; Khan K.M.; Farooq R.K.; Alomari M.; Islam I.; Algheribe S. |
Format: | Article |
Language: | English |
Published: |
Elsevier B.V.
2023
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Online Access: | https://www.scopus.com/inward/record.uri?eid=2-s2.0-85141287162&doi=10.1016%2fj.molstruc.2022.134449&partnerID=40&md5=31cc37b083234dc40107e9711af90b0d |
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