Synthesis, spectral analysis and biological evaluation of 2-{[(morpholin-4-yl)ethyl]thio}-5-phenyl/aryl-1,3,4-oxadiazole derivatives
A series of new derivatives of 4-(2-chloroethyl)morpholine hydrochloride (5) were efficiently synthesized. Briefly, different aromatic organic acids (1a-f) were refluxed to acquire respective esters (2a-f) using conc. H2SO4 as catalyst. The esters were subjected to nucleophillic substitution by mono...
Published in: | Pakistan Journal of Pharmaceutical Sciences |
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Main Author: | Aziz-Ur-Rehman; Khan S.G.; Naqvi S.A.R.; Ahmad M.; Akhtar N.; Bokhari T.H.; Irfan M.; Usman A.; Batool S.; Rasool S.; Shah S.A.A.; Shahid M. |
Format: | Article |
Language: | English |
Published: |
Pakistan Journal of Pharmaceutical Sciences
2021
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Online Access: | https://www.scopus.com/inward/record.uri?eid=2-s2.0-85107334212&doi=10.36721%2fPJPS.2021.34.1.SP.441-446.1&partnerID=40&md5=e8b212439da4fd6837b001731b079baa |
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