Convergent synthesis, free radical scavenging, Lineweaver-Burk plot exploration, hemolysis and in silico study of novel indole-phenyltriazole hybrid bearing acetamides as potent urease inhibitors

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Convergent synthesis, free radical scavenging, Lineweaver-Burk plot exploration, hemolysis and in silico study of novel indole-phenyltriazole hybrid bearing acetamides as potent urease inhibitors

In the current paper, through a convergent multi-step approach, a library of novel indole-phenyltriazole hybrids containing an amide moiety (9a-k) was synthesized. The structural verification of all synthesized molecules was accomplished by CHN and spectral analyses data. These synthesized bi-hetero...

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Bibliographic Details
Published in:	Journal of Heterocyclic Chemistry
Main Author:	Khan W.; Abbasi M.A.; Rehman A.-U.; Siddiqui S.Z.; Nazir M.; Ali Shah S.A.; Raza H.; Hassan M.; Shahid M.; Seo S.Y.
Format:	Article
Language:	English
Published:	HeteroCorporation 2020
Online Access:	https://www.scopus.com/inward/record.uri?eid=2-s2.0-85085113141&doi=10.1002%2fjhet.4006&partnerID=40&md5=f039d79804cdc8136fd9501b90993585

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