BSA Binding, molecular docking and in vitro biological screening of some new 1, 2, 4-triazole heterocycles bearing azinane nucleus

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BSA Binding, molecular docking and in vitro biological screening of some new 1, 2, 4-triazole heterocycles bearing azinane nucleus

A series of new compounds (5a-q), derived from 5-(1-(4-nitrophenylsulfonyl) piperidin-4-yl)-4-phenyl-4H-1,2,4-triazole-3-thiol (3) were proficiently synthesized to evaluate their biological activities. 1-(4-Nitrophenylsulfonyl) piperidine-4-carbohydrazide (2) was refluxed with phenylisothiocyanate t...

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Bibliographic Details
Published in:	Pakistan Journal of Pharmaceutical Sciences
Main Author:	Iqbal J.; Aziz-Ur-Rehman; Abbasi M.A.; Siddiqui S.Z.; Khalid H.; Laulloo S.J.; Chohan T.A.; Rasool S.; Ali Shah S.A.
Format:	Article
Language:	English
Published:	Pakistan Journal of Pharmaceutical Sciences 2020
Online Access:	https://www.scopus.com/inward/record.uri?eid=2-s2.0-85077920867&doi=10.36721%2fPJPS.2020.33.1.REG.149-160.1&partnerID=40&md5=5a5091bd9e7e9d2ef6cf1ce342b95d87

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