Synthesis, α-amylase inhibitory potential and molecular docking study of indole derivatives

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Synthesis, α-amylase inhibitory potential and molecular docking study of indole derivatives

In search of potent α-amylase inhibitor we have synthesized eighteen indole analogs (1–18), characterized by NMR and HR-EIMS and screened for α-amylase inhibitory activity. All analogs exhibited a variable degree of α-amylase inhibition with IC...

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Bibliographic Details
Published in:	Bioorganic Chemistry
Main Author:	Taha M.; Baharudin M.S.; Ismail N.H.; Imran S.; Khan M.N.; Rahim F.; Selvaraj M.; Chigurupati S.; Nawaz M.; Qureshi F.; Vijayabalan S.
Format:	Article
Language:	English
Published:	Academic Press Inc. 2018
Online Access:	https://www.scopus.com/inward/record.uri?eid=2-s2.0-85047793204&doi=10.1016%2fj.bioorg.2018.05.021&partnerID=40&md5=49c8b92a582bc139de13c9663d532f2a

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