Rational design of bis-indolylmethane-oxadiazole hybrids as inhibitors of thymidine phosphorylase

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Rational design of bis-indolylmethane-oxadiazole hybrids as inhibitors of thymidine phosphorylase

Inhibition of Thymidine phosphorylase (TP) is continuously studied for the design and development of new drugs for the treatment of neoplastic diseases. As a part of our effort to identify TP inhibitors, we performed a structure-based virtual screening (SBVS) of our compound collection. Based on the...

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Bibliographic Details
Published in:	Bioorganic and Medicinal Chemistry
Main Author:	Taha M.; Rashid U.; Imran S.; Ali M.
Format:	Article
Language:	English
Published:	Elsevier Ltd 2018
Online Access:	https://www.scopus.com/inward/record.uri?eid=2-s2.0-85047556645&doi=10.1016%2fj.bmc.2018.05.046&partnerID=40&md5=b8b86a9c07b0efb47642c7184ed60518

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