Synthesis: Small library of hybrid scaffolds of benzothiazole having hydrazone and evaluation of their β-glucuronidase activity

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Synthesis: Small library of hybrid scaffolds of benzothiazole having hydrazone and evaluation of their β-glucuronidase activity

Due to the great biological importance of β-glucuronidase inhibitors, here in this study, we have synthesized a library of novel benzothiazole derivatives (1–30), characterized by different spectroscopic methods and evaluated for β-glucuronidase inhibitory potential. Among the series sixteen compoun...

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Bibliographic Details
Published in:	Bioorganic Chemistry
Main Author:	Taha M.; Arbin M.; Ahmat N.; Imran S.; Rahim F.
Format:	Article
Language:	English
Published:	Academic Press Inc. 2018
Online Access:	https://www.scopus.com/inward/record.uri?eid=2-s2.0-85040336943&doi=10.1016%2fj.bioorg.2018.01.002&partnerID=40&md5=9227c9c6d5b8595109fb377272a53c00

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