Synthesis and structural analysis of persuasive antibacterial agents and enzyme inhibitors derived from 5-(1-(4-Tosyl)piperidin-4-yl)-1,3,4-oxadiazol-2-thiol

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Synthesis and structural analysis of persuasive antibacterial agents and enzyme inhibitors derived from 5-(1-(4-Tosyl)piperidin-4-yl)-1,3,4-oxadiazol-2-thiol

Due to outstanding biological activities of 1,3,4-oxadiazole, a series of S-substituted derivatives of 5-[1-(4-tosyl)piperidin-4-yl]-1,3,4-oxadiazol-2-thiol (5a-f) was synthesized. The reaction of p-toluene sulfonyl chloride (a) with ethyl isonepacotate (b) produced ethyl 1-(4-tosyl)piperidin-4-carb...

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Bibliographic Details
Published in:	Asian Journal of Chemistry
Main Author:	Aziz-Ur-Rehman; Sattar A.; Abbasi M.A.; Siddiqui S.Z.; Raza M.A.; Ashraf M.; Nazir M.; Shah S.A.A.
Format:	Article
Language:	English
Published:	Chemical Publishing Co. 2018
Online Access:	https://www.scopus.com/inward/record.uri?eid=2-s2.0-85040132566&doi=10.14233%2fajchem.2018.20871&partnerID=40&md5=157c83646ac804918a4b607e79e83dff

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